研究業績 (学会発表 2011年度)
Preclinical validation of the sensitivity and specificity of a fluorescent nanobeacon for its application in colonoscopy-based imaging of colorectal cancer
Wellington Pham, Hironori Kumagai, Ken-Ichiro Hiwatari, Hiroyuki Tachikawa, Ryoji Kimura, Kunio Nakamura, Makoto Kataoka, Shinji Yamashita, Shinji Sakuma
AACR 102nd Annual Meeting 2011
Orlando, FL
20110405

Lectin-immobilized fluorescent nanospheres as a diagnostic agent for colonoscopy
片岡 誠東野 晴輝押谷 仁美政岡 祥江山下 伸二、日渡 謙一郎、立川 裕之、木村 凌治、中村 邦生、Huaiyu Ma、Zhijian Yang、Li Tang、Robert M. Hoffman、熊谷 光倫、John C Gore、Wellington Pham、佐久間 信至
第6回日本分子イメージング学会
神戸
20110526

胃内薬物溶解を考慮した難溶解性薬物の経口吸収性評価システムの構築
深堀 美秀片岡 誠政岡 祥江佐久間 信至山下 伸二
日本薬剤学会第26年会
東京
20110529

コア-シェル型ナノ粒子化による難水溶性薬物の経口吸収改善
山本 真梨奈佐久間 信至政岡 祥江片岡 誠山下 伸二、張 紹玲、 川上 亘作
日本薬剤学会第26年会
東京
20110529

レクチン固定化ナノバイオコンジュゲートの糖鎖認識能の検証
押谷 仁美佐久間 信至政岡 祥江片岡 誠山下 伸二、日渡 謙一郎、 立川 裕之、 木村 凌治、 中村 邦生、 熊谷 光倫、John C.Gore、 Wellington Pham
日本薬剤学会第26年会
東京
20110529

Positron emission tomographyを用いたテルミサルタン経口投与後の体内動態評価
片岡 誠、 高島 忠之、 新垣 友隆、 政岡 祥江佐久間 信至、片山 由美子、 橋爪 良信、 和田 康弘、 杉山 雄一、 渡辺 恭良、山下 伸二
日本薬剤学会第26年会
東京
20110531

D/Pシステムを用いた胃での溶解過程を含む経口吸収性評価系の構築
竹山 匠子、 新垣 友隆、 徳田 英昭、 古市 丈治、 李 英培、片岡 誠山下 伸二
日本薬剤学会第26年会
東京
20110531

デンドリマー型アルブチンの化学構造とSGLT1(Na+/糖共輸送体)の阻害活性との相関の検証
金光 俊佐久間 信至寺岡 裕美山下 伸二、白坂 善之、玉井 郁巳、村岡 雅弘、中辻 洋司、木田 敏之、明石 満
第27会日本DDS学会学術集会
東京
20110609

粘膜投与型ワクチンの抗原キャリアとしてのオリゴアルギニン固定化高分子の可能性評価
井上 咲姫佐久間 信至吹田 正哉政岡 祥江片岡 誠山下 伸二、山内 仁史、日渡 謙一郎、宇都 倫史、馬場 昌範
第27会日本DDS学会学術集会
東京
20110610

IVIVC consideration based on the analysis of in vivo oral absorption process in human
S. Yamashita
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Evaluation of oral absorption of basic drugs with poor water-solubility using in vitro dissolution/permeation system: effect of drug dissolution in the stomach.
Miho Fukahori, Makoto Kataoka, Yoshie Masaoka, Shinji Sakuma, Shinji Yamashita.
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

A potential of oligoarginine-linked polymers as carriers for mucosal delivery of vaccines.
Saki Inoue, Shinji Sakuma, Masaya Suita, Yoshie Masaoka, Makoto Kataoka, Shinji Yamashita, Noriko Nakajima, Norihiro Shinkai, Hitoshi Yamauchi, Ken-Ichiro Hiwatari, Hiroyuki Tachikawa, Ryouji Kimura, Tomofumi Uto, Masanori Baba
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Enhancement of oral absorption of poorly water-soluble drugs through core-shell-structured formulations.
Marina Yamamoto, Shinji Sakuma, Yoshie Masaoka, Makoto Kataoka, Shinji Yamashita, Shaoling Zhang, Kohsaku Kawakami
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Effect of meglumine on the dissolution and precipitation of telmisartan in the GI tract.
Arima Fukunishi, Makoto Kataoka, Koichi Wada, Shinji Yamashita
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Advanced strategy for the practical use of in vitro dissolution/permeation system in the development of oral drug products.
Shoko Takeyama, Tomotaka Shingaki, Hideaki Tokuda, Joji Furuichi, Eibai Lee, Makoto Kataoka, Shinji Yamashita
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Imaging of gastrointestinal absorption process of orally administered drugs using positron emission tomography.
Makoto Kataoka, Tadayuki Takashima, Tomotaka Shingaki, Yoshie Masaoka, Shinji Sakuma, Yumiko Katayama, Emi Hayashinaka, Yasuhiro Wada, Yilong Cui, Yasuyoshi Watanabe, Shinji Yamashita
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Positron emission tomography study of gastrointestinal absorption process of [11C]telmisartan after oral administration.
Tadayuki Takashima, Makoto Kataoka, Tomotaka Shingaki, Yumiko Katayama, Yoshinobu Hashizume, Hiroyuki Ou, Yasuhiro Wada, Shinji Yamashita, Yasuyoshi Watanabe
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Optimization of surface structure of peanut agglutinin-immobilized nanospheres as a colonoscopic imaging agent.
Hitomi Oshitani, Shinji Sakuma, Yoshie Masaoka, Makoto Kataoka, Shinji Yamashita, Ken-Ichiro Hiwatari, Hiroyuki Tachikawa, Ryoji Kimura, Kunio Nakamura, Hironori Kumagai, John C. Gore, Wellington Pham
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Essence of affinity and specificity of lectin-immobilized fluorescent nanospheres for colonic tumors.
Haruki Higashino, Shinji Sakuma, Yoshie Masaoka, Makoto Kataoka, Shinji Yamashita, Ken-Ichiro Hiwatari, Hiroyuki Tachikawa, Ryoji Kimura, Kunio Nakamura, Hironori Kumagai, John C. Gore, Wellington Pham
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Inhibitory effect of arbutin conjugated to polyamidoamine dendrimers on intestinal glucose transport.
Shun Kanamitsu, Shinji Sakuma, Yumi Teraoka, Yoshie Masaoka, Makoto Kataoka, Shinji Yamashita, Yoshiyuki Shirasaka, Ikumi Tamai, Masahiro Muraoka, Yohji Nakatsuji, Toshiyuki Kida, Mitsuru Akashi
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Elucidation of intestinal absorption mechanism of 2-fluoro-2-deoxy-D-glucose.
Ryutarou Katagiri, Makoto Kataoka, Yoshie Masaoka, Shinji Sakuma, Shinji Yamashita
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Effect of supersaturation on oral absorption of poorly water-soluble drugs: dissolution/permeation system with rat small intestine.
Kanami Nishi, Makoto Kataoka, Yoshie Masaoka, Shinji Sakuma, Shinji Yamashita
International Symposium on BA/BE of Oral Drug Products: More Science, Technology and Better Regulatory Standards
Kobe
20110630

Peanut Agglutinin-immobilized Fluorescent Nanospheres with Surface Poly(N-vinylacetamide) Chains as a Safe Candidate of Diagnostic Drugs for Colonoscopy
M. Kataoka, S. Sakuma, H. Higashino, T. Yano, Y. Masaoka, S. Yamashita, K. Hiwatari, H. Tachikawa, R.Kimura, K. Nakamura, H. Kumagai, J.C. Gore, W. Pham
38th Annual Meeting & Exposition of the Controlled Release Society
National Harbor MD
20110802

Use of Positron Emission Tomography for the Analysis of Gastrointestinal Drug Absorption in Human
Tadayuki Takashima, Tomotaka Shingaki, Masaaki Tanaka, Yoshihito Shigihara, Yasuhiro Wada, Makoto Kataoka, Yuichi Sugiyama, Shinji Yamashita, Yasuyoshi Watanabe
World Molecular Imaging Congress 2011
San Diego, CA
20110907

薬物動態研究への分子イメージング技術の利用―PETを用いた経口吸収過程の解析―
片岡 誠、高島 忠之、新垣 友隆、和田 康弘、政岡 祥江佐久間 信至、渡辺 恭良、山下 伸二
第61回日本薬学会近畿支部総会・大会
神戸
20111022

Quantitative Analysis of the effect of Supersaturation on in Vivo Drug Absorption
Shinji Yamashita
2011 American Association of Pharmaceutical Scientists (AAPS) Annual Meeting and Exposition
Washington, DC
20111024

EFFECT OF SUPERSATURATION ON ORAL ABSORPTION OF POORLY WATER-SOLUBLE DRUGS: IN VITRO ASSESSMENT USING DISSOLUTION/PERMEATION SYSTEM
Makoto Kataoka, Ryusuke Takano, Kentaro Furumoto, Shinichi Yoshizaki, Nozomi Hisada, Yoshie Masaoka, Shinji Sakuma, Shinji Yamashita
26th JSSX Annual Meeting
Hiroshima
20111117

QUANTIFICATION OF SPECIES DIFFERENCES IN THE EFFECT OF P-GLYCOPROTEIN ON INTESTINAL DRUG ABSORPTION
Haruki Higashino, Samantha K. Mathur, Yoshiki Katada, Yoshie Masaoka, Makoto Kataoka, Shinji Sakuma, Shinji Yamashita
26th JSSX Annual Meeting
Hiroshima
20111118

INNOVATIVE STRATEGIES FOR DRUG DEVELOPMENT USING MICRODOSING CLINICAL STUDIES (NEDO MICRODOSE-PJ) 2011 (7): DEVELOPMENT OF ORAL FORMULATIONS FOR MD STUDY
Yoshie Masaoka, Makoto Kataoka, Shinji Sakuma, Yuki Suzaki, Hiromitsu Imai, Tsutomu Kotegawa, Takuya Morimoto, Kyoichi Ohashi, Yuichi Sugiyama, Shinji Yamashita
26th JSSX Annual Meeting
Hiroshima
20111118

Impact of BCS on Development and Quality Control of Oral Drug Product
Shinji Yamashita
Asian Federation for Pharmaceutical Sciences Conference 2011
Kuala Lumpur
20111210

Development of oral formulations for MD study
Yoshie Masaoka, Makoto Kataoka, Shinji Sakuma, Yuki Suzaki, Hiromitsu Imai, Tsutomu Kotegawa, Takuya Morimoto, Kyoichi Ohashi, Yuichi Sugiyama, Shinji Yamashita
PPF Molecular Pharmacokinetics
Tokyo
20120116

Effect of P-glycoprotein-mediated efflux on oral drug absorption: in vitro assessment with dissolution/permeation system
Makoto Kataoka, Yoshie Masaoka, Shinji Sakuma, Shinji Yamashita
PPF Molecular Pharmacokinetics
Tokyo
20120117

Prediction of oral drug absorption in human based on dissolution and permeation profiles in GI tract
Shinji Yamashita
PPF Molecular Pharmacokinetics
Tokyo
20120118

Design of nanoparticulate solid dispersions using electrospray deposition
Kohsaku Kawakami, Shaoling Zhang, Marina Yamamoto, Yoshie Masaoka, Makoto Kataoka, Shinji Yamashita, Shinji Sakuma
8th World Meeting on Pharmaceutics, Biopharmaceutics and Pharmaceutical Technology
Istanbul
20120319

薬剤師の生涯教育における摂南大学薬学部の取り組み
山口 昌之、吉岡 靖啓、首藤 誠、荻田 喜代一、佐久間 信至、前田 定秋
日本薬学会第132年会
札幌
20120329

BCSコンセプトに基づくヒト同等性試験におけるリスクファクターの解析
山下 伸二佐久間 信至
日本薬学会第132年会
札幌
20120329

Dissolution/permeationシステムを用いた難溶解性薬物の経口投与製剤スクリーニング
片岡 誠、Kiyohiko Sugano、Claudia da Costa Mathews、Jing-Wen Wong、Kelly Lane Jones、政岡 祥江佐久間 信至山下 伸二
日本薬学会第132年会
札幌
20120330

消化管膜機能制御に基づく抗糖尿病作用を有する配糖体―高分子複合体の精密設計
佐久間 信至金光 俊寺岡 裕美政岡 祥江片岡 誠山下 伸二、白坂 善之、玉井 郁巳、村岡 雅弘、中辻 洋司、木田 敏之、明石 満
日本薬学会第132年会
札幌
20120330